Regioselective 1,4-conjugate aza-Michael addition of dienones with benzotriazole-Reference-Cited by-同舟云学术

Regioselective 1,4-conjugate aza-Michael addition of dienones with benzotriazole

Published:2017-01-01 Issue:4 Volume:23 Page:
ISSN:2191-0197
Container-title:Heterocyclic Communications
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Author:

Li Zheng,Li Tianpeng,Fu Rugang,Yang Jingya

Abstract

AbstractThe regioselective 1,4-conjugate aza-Michael addition of dienones with benzotriazole catalyzed by potassium acetate is described. A series of 3-(benzotriazol-1-yl)-1,5-diarylpent-4-en-1-ones were efficiently synthesized under mild conditions. This protocol has advantages of transition-metal free catalyst, high yield and high regioselectivity.

Publisher

Walter de Gruyter GmbH

Subject

Organic Chemistry

Link

https://www.degruyter.com/document/doi/10.1515/hc-2016-0182/pdf

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