Synthesis and Biological Evaluation of 3,9-Dioxatetraasteranes as C2-Symmetric HIV-1 Protease Inhibitors and Docking Study
Author:
Affiliation:
1. Beijing Key Laboratory of Environmental and Viral Oncology, College of Life Science and Bioengineering, Beijing University of Technology
Publisher
Pharmaceutical Society of Japan
Subject
Pharmaceutical Science,Pharmacology,General Medicine
Link
https://www.jstage.jst.go.jp/article/bpb/42/2/42_b18-00705/_pdf
Reference16 articles.
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3. 3) Huff JR, Kahn J. Discovery and clinical development of HIV-1 protease inhibitors. Adv. Protein Chem., 56, 213–251 (2001).
4. 4) Brik A, Wong C-H. HIV-1 protease: mechanism and drug discovery. Org. Biomol. Chem., 1, 5–14 (2003).
5. 5) Greer J, Erickson JW, Baldwin JJ, Varney MD. Application of the three-dimensional structures of protein target molecules in structure-based drug design. J. Med. Chem., 37, 1035–1054 (1994).
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