Clastogenicity of Quinoline Derivatives in the Liver Micronucleus Assay Using Rats and Mice

Author:

Hakura Atsushi1,Kadoi Minoru2,Suzuki Takayoshi3,Saeki Ken-ichi2

Affiliation:

1. Drug Safety Research Laboratories, Eisai Co., Ltd.

2. Graduate School of Pharmaceutical Sciences, Nagoya City University

3. Division of Cellular and Gene Therapy Products, National Institute of Health Sciences

Publisher

Pharmaceutical Society of Japan

Subject

Health, Toxicology and Mutagenesis,Toxicology

Reference17 articles.

1. Modification of the Carcinogenic Potency of Quinoline, a Hepatocarcinogen, by Fluorine Atom Substitution: Evaluation of Carcinogenicity by a Medium-Term Assay.

2. 2) Hirao, N., Shinohara, Y., Tsuda, H., Fukushima, S., Takahashi, M. and Ito, N. (1976) Carcinogenic activity of quinoline on rat liver. Cancer Res., 36, 329-335.

3. 3) Shinohara, Y., Ogiso, T., Hananouchi, M., Nakanishi, K., Yoshimura, T. and Ito, N. (1977) Effects of various factors on the induction of liver tumors in animals by quinoline. Jpn. J. Cancer Res., 68, 785-796.

4. 4) Wayand, E. H., Defauw, J., McQueen, C. A., Meschter, C. L., Meegalla, S. K. and LaVoie, E. J. (1993) Bioassay of quinoline, 5-fluoroquinoline, carbazole, 9-methylcarbazole and 9-ethylcarbazole in newborn mice. Food Chem. Toxicol., 31, 707-715.

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