Rational design and synthesis of a novel class of active site-targeted HIV protease inhibitors containing a hydroxymethylcarbonyl isostere. Use of phenylnorstatine or allophenylnorstatine as a transition-state mimic.-Reference-Cited by-同舟云学术

Rational design and synthesis of a novel class of active site-targeted HIV protease inhibitors containing a hydroxymethylcarbonyl isostere. Use of phenylnorstatine or allophenylnorstatine as a transition-state mimic.

Published:1991 Issue:9 Volume:39 Page:2465-2467
ISSN:0009-2363
Container-title:Chemical and Pharmaceutical Bulletin
language:en
Short-container-title:CHEMICAL & PHARMACEUTICAL BULLETIN

Author:

MIMOTO Tsutomu,IMAI Junya,TANAKA Shigeki,HATTORI Naoko,TAKAHASHI Osamu,KISANUKI Sumitsugu,NAGANO Yuichi,SHINTANI Makoto,HAYASHI Hideya,SAKIKAWA Hiroshi,AKAJI Kenichi,KISO Yoshiaki

Publisher

Pharmaceutical Society of Japan

Subject

Drug Discovery,General Chemistry,General Medicine

Link

http://www.jstage.jst.go.jp/article/cpb1958/39/9/39_9_2465/_pdf

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