Development of Sarpogrelate External Preparation for Intractable Pain Control. I. Pre-formulation Study on Application of Modified .BETA.-Cyclodextrins-Reference-Cited by-同舟云学术

Development of Sarpogrelate External Preparation for Intractable Pain Control. I. Pre-formulation Study on Application of Modified .BETA.-Cyclodextrins

Published:2010 Issue:1 Volume:58 Page:45-50
ISSN:0009-2363
Container-title:Chemical and Pharmaceutical Bulletin
language:en
Short-container-title:CHEMICAL & PHARMACEUTICAL BULLETIN

Author:

Hanawa Kazumi¹²,Hanawa Takehisa¹,Tsuchiya Chikako¹,Higashi Kenjirou²,Suzuki Masahiko¹,Moribe Kunikazu²,Yamamoto Keiji²,Oguchi Toshio¹

Affiliation:

1. Department of Pharmacy, University Hospital, University of Yamanashi

2. Graduate School of Pharmaceutical Sciences, Chiba University

Publisher

Pharmaceutical Society of Japan

Subject

Drug Discovery,General Chemistry,General Medicine

Link

http://www.jstage.jst.go.jp/article/cpb/58/1/58_1_45/_pdf

Reference20 articles.

1. Effects of a 5-HT2A receptor antagonist, sarpogrelate on thermal or inflammatory pain

2. Peripheral 5-HT2A receptor antagonism attenuates primary thermal hyperalgesia and secondary mechanical allodynia after thermal injury in rats

3. Sarpogrelate Hydrochloride, a 5-HT2A Receptor Antagonist, Attenuates Neurogenic Pain Induced by Nucleus Pulposus in Rats

4. Topical ketanserin attenuates hyperalgesia and inflammation in arthritis in rats

5. 5) Serata K., Ikeda T., Iida Y., Okuni H., Tomaru T., Serotonin(5-HT2) Kenkyukai Houkoku, 34—35 (1997).

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