cAMP Signaling Pathway Prevents Dasatinib-Induced Vascular Hyperpermeability

Author:

Aoyama Tsuyoshi1,Kuriyama Hiroki1,Sato Yuki1,Imai Shungo1,Kashiwagi Hitoshi1,Sugawara Mitsuru1,Takekuma Yoh2

Affiliation:

1. Laboratory of Pharmacokinetics, Faculty of Pharmaceutical Sciences, Hokkaido University

2. Department of Pharmacy, Hokkaido University Hospital

Publisher

Pharmaceutical Society of Japan

Subject

Pharmaceutical Science,Pharmacology,General Medicine

Reference38 articles.

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2. 2) Nakamae H, Fukuda T, Nakaseko C, Kanda Y, Ohmine K, Ono T, Matsumura I, Matsuda A, Aoki M, Ito K, Shibayama H. Nilotinib vs. imatinib in Japanese patients with newly diagnosed chronic myeloid leukemia in chronic phase: long-term follow-up of the Japanese subgroup of the randomized ENESTnd trial. Int. J. Hematol., 107, 327–336 (2018).

3. 3) Miura M. Therapeutic drug monitoring of imatinib, nilotinib, and dasatinib for patients with chronic myeloid leukemia. Biol. Pharm. Bull., 38, 645–654 (2015).

4. 4) Riou M, Seferian A, Savale L, Chaumais MC, Guignabert C, Canuet M, Magro P, Rea D, Sitbon O, Jaïs X, Humbert M, Montani D. Deterioration of pulmonary hypertension and pleural effusion with bosutinib following dasatinib lung toxicity. Eur. Respir. J., 48, 1517–1519 (2016).

5. 5) Kantarjian H, Shah NP, Hochhaus A, Cortes J, Shah S, Ayala M, Moiraghi B, Shen Z, Mayer J, Pasquini R, Nakamae H, Huguet F, Boqué C, Chuah C, Bleickardt E, Bradley-Garelik MB, Zhu C, Szatrowski T, Shapiro D, Baccarani M. Dasatinib versus imatinib in newly diagnosed chronic-phase chronic myeloid leukemia. N. Engl. J. Med., 362, 2260–2270 (2010).

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