Effects of Bepridil and Pimozide, Existing Medicines Capable of Blocking T-Type Ca<sup>2+</sup> Channels, on Visceral Pain in Mice-Reference-Cited by-同舟云学术

Effects of Bepridil and Pimozide, Existing Medicines Capable of Blocking T-Type Ca²⁺ Channels, on Visceral Pain in Mice

Published:2021-03-01 Issue:3 Volume:44 Page:461-464
ISSN:0918-6158
Container-title:Biological and Pharmaceutical Bulletin
language:en
Short-container-title:Biol. Pharm. Bull.

Author:

Tsubota Maho¹,Matsui Kazuki¹,Fukushi Saaya¹,Okazaki Kyoko¹,Sekiguchi Fumiko¹,Kawabata Atsufumi¹

Affiliation:

1. Laboratory of Pharmacology and Pathophysiology, Faculty of Pharmacy, Kindai University

Publisher

Pharmaceutical Society of Japan

Subject

Pharmaceutical Science,Pharmacology,General Medicine

Link

https://www.jstage.jst.go.jp/article/bpb/44/3/44_b20-00742/_pdf

Reference23 articles.

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2. 2) Weiss N, Zamponi GW. T-type calcium channels: from molecule to therapeutic opportunities. Int. J. Biochem. Cell Biol., 108, 34–39 (2019).

3. 3) Snutch TP, Zamponi GW. Recent advances in the development of T-type calcium channel blockers for pain intervention. Br. J. Pharmacol., 175, 2375–2383 (2018).

4. 4) Uchino T, Lee TS, Kaku T, Yamashita N, Noguchi T, Ono K. Voltage-dependent and frequency-independent inhibition of recombinant Ca_v3.2 T-type Ca²⁺ channel by bepridil. Pharmacology, 74, 174–181 (2005).

5. 5) Santi CM, Cayabyab FS, Sutton KG, McRory JE, Mezeyova J, Hamming KS, Parker D, Stea A, Snutch TP. Differential inhibition of T-type calcium channels by neuroleptics. J. Neurosci., 22, 396–403 (2002).

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