Anti-allodynic and Neuroprotective Effects of Koumine, a Benth Alkaloid, in a Rat Model of Diabetic Neuropathy

Author:

Ling Qian1,Liu Ming1,Wu Min-Xia1,Xu Ying1,Yang Jian1,Huang Hui-Hui1,Yu Chang-Xi1

Affiliation:

1. Department of Pharmacology, College of Pharmacy, Fujian Medical University

Publisher

Pharmaceutical Society of Japan

Subject

Pharmaceutical Science,Pharmacology,General Medicine

Reference20 articles.

1. 1) Edwards JL, Vincent AM, Cheng HT, Feldman EL. Diabetic neuropathy: mechanisms to management. Pharmacol. Ther., 120, 1–34 (2008).

2. 2) Dworkin RH, O’Connor AB, Backonja M, Farrar JT, Finnerup NB, Jensen TS, Kalso EA, Loeser JD, Miaskowski C, Nurmikko TJ, Portenoy RK, Rice AS, Stacey BR, Treede RD, Turk DC, Wallace MS. Pharmacologic management of neuropathic pain: evidence-based recommendations. Pain, 132, 237–251 (2007).

3. 3) Tomlinson DR, Gardiner NJ. Glucose neurotoxicity. Nat. Rev. Neurosci., 9, 36–45 (2008).

4. 4) Xu Y, Qiu HQ, Liu H, Liu M, Huang ZY, Yang J, Su YP, Yu CX. Effects of koumine, an alkaloid of Gelsemium elegans BENTH., on inflammatory and neuropathic pain models and possible mechanism with allopregnanolone. Pharmacol. Biochem. Behav., 101, 504–514 (2012).

5. 5) Su YP, Shen J, Xu Y, Zheng M, Yu CX. Preparative separation of alkaloids from Gelsemium elegans BENTH. using pH-zone-refining counter-current chromatography. J. Chromatogr. A, 1218, 3695–3698 (2011).

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