Advances in predicting CYP-mediated drug interactions in the drug discovery setting
Author:
Publisher
Informa Healthcare
Subject
Drug Discovery
Link
http://www.tandfonline.com/doi/pdf/10.1517/17460441.1.7.677
Reference124 articles.
1. Can the pharmaceutical industry reduce attrition rates?
2. High-Throughput Screening in Drug Metabolism and Pharmacokinetic Support of Drug Discovery
3. Automated high throughput ADME assays for metabolic stability and cytochrome P450 inhibition profiling of combinatorial libraries
4. Do Drug Metabolism and Pharmacokinetic Departments Make Any Contribution to Drug Discovery?
5. Characteristics and common properties of inhibitors, inducers, and activators of CYP enzymes
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2. Mechanisms of promiscuity among drug metabolizing enzymes and drug transporters;The FEBS Journal;2019-11-12
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5. Evaluation of CYP2C8 Inhibition In Vitro: Utility of Montelukast as a Selective CYP2C8 Probe Substrate;Drug Metabolism and Disposition;2011-06-22
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