Drug design and development through the vanilloid receptor
Author:
Affiliation:
1. Centro de Investigación Príncipe Felipe, Valencia, Spain
2. Universidad Miguel Hernández, Instituto Biología Molecular y Celular, Ed. Torregaitan, Av. De la Universidad s/n, 03202 Elche, Alicante, Spain ; ;
Publisher
Informa Healthcare
Subject
Drug Discovery
Link
https://www.tandfonline.com/doi/pdf/10.1517/17460441.2.8.1053
Reference87 articles.
1. Molecular mechanisms of nociception
2. The Vanilloid Receptor: A Molecular Gateway to the Pain Pathway
3. Transient Receptor Potential Cation Channels in Disease
4. The vanilloid receptor TRPV1: 10 years from channel cloning to antagonist proof-of-concept
5. The Vanilloid Receptor TRPV1 Is Tonically Activated In Vivo and Involved in Body Temperature Regulation
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2. Adamantyl Analogues of Paracetamol as Potent Analgesic Drugs via Inhibition of TRPA1;PLoS ONE;2014-12-01
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4. N-Pyridin-3-yl- and N-quinolin-3-yl-benzamides: Modulators of Human Vanilloid Receptor 1 (TRPV1);Bioorganic & Medicinal Chemistry Letters;2008-04
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