Radioligand dissociation measurements: potential interference of rebinding and allosteric mechanisms and physiological relevance of the biological model systems-Reference-Cited by-同舟云学术

Radioligand dissociation measurements: potential interference of rebinding and allosteric mechanisms and physiological relevance of the biological model systems

Published:2012-06 Issue:7 Volume:7 Page:583-595
ISSN:1746-0441
Container-title:Expert Opinion on Drug Discovery
language:en
Short-container-title:Expert Opinion on Drug Discovery

Author:

Vauquelin Georges,Van Liefde Isabelle

Publisher

Informa UK Limited

Subject

Drug Discovery

Link

http://www.tandfonline.com/doi/pdf/10.1517/17460441.2012.687720

Reference100 articles.

1. Kinetics of pharmacologic response

2. Association of Candesartan vs Losartan With All-Cause Mortality in Patients With Heart Failure

3. Effects of losartan vs candesartan in reducing cardiovascular events in the primary treatment of hypertension

4. Biochemical mechanisms of drug action: what does it take for success?

5. Biochemical Mechanisms of New Molecular Entities (NMEs) Approved by United States FDA During 2001-2004: Mechanisms Leading to Optimal Efficacy and Safety

Cited by 22 articles. 订阅此论文施引文献订阅此论文施引文献，注册后可以免费订阅5篇论文的施引文献，订阅后可以查看论文全部施引文献

1. Probe dependency in the determination of ligand binding kinetics at a prototypical G protein-coupled receptor;Scientific Reports;2019-05-27

2. Binding kinetics of ligands acting at GPCRs;Molecular and Cellular Endocrinology;2019-04

3. Assays with Detection of Fluorescence Anisotropy: Challenges and Possibilities for Characterizing Ligand Binding to GPCRs;Trends in Pharmacological Sciences;2018-02

4. Drug target residence time: a misleading concept;Drug Discovery Today;2018-01

5. Competitive ligands facilitate dissociation of the complex of bifunctional inhibitor and protein kinase;Biophysical Chemistry;2017-09