Design, synthesis and biological evaluation of dipeptides as novel non-covalent 20S proteasome inhibitors-Reference-Cited by-同舟云学术

Design, synthesis and biological evaluation of dipeptides as novel non-covalent 20S proteasome inhibitors

Published:2021-04-12 Issue:5 Volume:23 Page:436-451
ISSN:1028-6020
Container-title:Journal of Asian Natural Products Research
language:en
Short-container-title:Journal of Asian Natural Products Research

Author:

Yang Ya-Jun¹,Wang Ke¹,Yang Ying¹,Lai Fang-Fang²,Chen Xiao-Guang²,Xiao Zhi-Yan¹

Affiliation:

1. Beijing Key Laboratory of Active Substance Discovery and Druggability Evaluation, Institute of Materia Medica, Chinese Academy of Medical Sciences and Peking Union Medical College, Beijing 100050, China

2. The State Key Laboratory of Bioactive Substance and Function of Natural Medicines, Institute of Material Medica, Chinese Academy of Medical Sciences and Peking Union Medical College, Beijing 100050, China

Funder

National Natural Science Foundation of China

the CAMS Innovation Fund for Medical Sciences

Publisher

Informa UK Limited

Subject

Organic Chemistry,Complementary and alternative medicine,Drug Discovery,Pharmaceutical Science,Pharmacology,Molecular Medicine,General Medicine,Analytical Chemistry

Link

https://www.tandfonline.com/doi/pdf/10.1080/10286020.2021.1910241

Reference21 articles.

1. Recognition and Processing of Ubiquitin-Protein Conjugates by the Proteasome

2. Synthesis and Pharmacology of Proteasome Inhibitors

3. Proteasome Inhibitors: Recent Advances and New Perspectives In Medicinal Chemistry

4. The Proteasome: Paradigm of a Self-Compartmentalizing Protease

5. Importance of the Different Proteolytic Sites of the Proteasome and the Efficacy of Inhibitors Varies with the Protein Substrate

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1. Design, synthesis, and biological evaluation of some novel naphthoquinone‐glycine/β‐alanine anilide derivatives as noncovalent proteasome inhibitors;Chemical Biology & Drug Design;2023-02-17

2. Fungal Secondary Metabolites as Inhibitors of the Ubiquitin–Proteasome System;International Journal of Molecular Sciences;2021-12-10