Synthesis and Biological Evaluation of Novel N-[3-fluoro-4-(morpholin-4-yl)phenyl]thiazol-2-amine Derivatives as Potent Antibacterial and Anticancer Agents and ADMET-Reference-Cited by-同舟云学术

Synthesis and Biological Evaluation of Novel N-[3-fluoro-4-(morpholin-4-yl)phenyl]thiazol-2-amine Derivatives as Potent Antibacterial and Anticancer Agents and ADMET

Published:2023-01-25 Issue:1 Volume:44 Page:117-128
ISSN:1040-6638
Container-title:Polycyclic Aromatic Compounds
language:en
Short-container-title:Polycyclic Aromatic Compounds

Author:

Nellutla Manoj Kumar¹²,Kamarajugadda Pavan²,Soma Laxminarayana²,Haridasyam Ramesh Babu³,Narsimha Sirassu¹^ORCID

Affiliation:

1. Department of Chemistry, Chaitanya (Deemed to be University), Hanamkonda, India

2. Aragen Life Sciences, Hyderabad, India

3. Department of Physical Sciences/Chemistry, Kakatiya Institute of Technology and Science, Hanumakonda, India

Publisher

Informa UK Limited

Subject

Materials Chemistry,Organic Chemistry,Polymers and Plastics

Link

https://www.tandfonline.com/doi/pdf/10.1080/10406638.2023.2169473

Reference32 articles.

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2. Benzothiazoles exhibit broad-spectrum antitumor activity: Their potency, structure–activity and structure–metabolism relationships

3. Immune checkpoint inhibitors: a promising anticancer therapy

4. Synthesis, cytotoxicity and antimicrobial activity of thiourea derivatives incorporating 3-(trifluoromethyl)phenyl moiety

5. Inhibitors of antibiotic resistance mechanisms: clinical applications and future perspectives

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