Dihydrofolate reductase inhibitors: patent landscape and phases of clinical development (2001

Dihydrofolate reductase inhibitors: patent landscape and phases of clinical development (2001–2021)

Published:2022-10-03 Issue:10 Volume:32 Page:1079-1095
ISSN:1354-3776
Container-title:Expert Opinion on Therapeutic Patents
language:en
Short-container-title:Expert Opinion on Therapeutic Patents

Author:

Bhagat Kavita¹²^ORCID,Kumar Nitish¹^ORCID,Kaur Gulati Harmandeep¹,Sharma Aanchal¹,Kaur Amandeep¹,Singh Jatinder Vir¹,Singh Harbinder¹,Bedi Preet Mohinder Singh¹^ORCID

Affiliation:

1. Department of Pharmaceutical Sciences, Guru Nanak Dev University, Amritsar, India

2. Department of Pharmaceutical Sciences, Khalsa College of Pharmacy, Amritsar, India

Funder

Department of Science and Technology

Publisher

Informa UK Limited

Subject

Drug Discovery,Pharmacology,General Medicine

Link

https://www.tandfonline.com/doi/pdf/10.1080/13543776.2022.2130752

Reference79 articles.

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2. Structural comparison of chromosomal and exogenous dihydrofolate reductase fromStaphylococcus aureusin complex with the potent inhibitor trimethoprim

3. The identification of novel Mycobacterium tuberculosis DHFR inhibitors and the investigation of their binding preferences by using molecular modelling

4. Chemical space ofEscherichia colidihydrofolate reductase inhibitors: New approaches for discovering novel drugs for old bugs

5. Effectiveness of Antimalarial Drugs

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