A novel chromone-based as a potential inhibitor of ULK1 that modulates autophagy and induces apoptosis in colon cancer

Author:

Shamsudin Nur Farisya1,Leong Sze-Wei2,Koeberle Andreas3,Suriya Utid4,Rungrotmongkol Thanyada4,Chia Suet Lin5,Taher Muhammad6,Haris Muhammad Salahuddin6,Alshwyeh Hussah Abdullah78,Alosaimi Areej A8,Mediani Ahmed9,Ilowefah Muna Abdulsalam10,Islami Deri11,Mohd Faudzi Siti Munirah12,Fasihi Mohd Aluwi Mohd Fadhlizil13,Wai Lam Kok14,Rullah Kamal1ORCID

Affiliation:

1. Drug Discovery & Synthetic Chemistry Research Group, Department of Pharmaceutical Chemistry, Kulliyyah of Pharmacy, International Islamic University Malaysia, Bandar Indera Mahkota, Kuantan 25200, Pahang, Malaysia

2. Department of Chemistry, Faculty of Science, University of Malaya, Kuala Lumpur 50603, Malaysia

3. Michael Popp Institute & Center for Molecular Biosciences Innsbruck (CMBI), University of Innsbruck, Innsbruck 6020, Austria

4. Structural & Computational Biology Research Unit, Department of Biochemistry, Faculty of Science, Chulalongkorn University, Bangkok 10330, Thailand

5. UPM – MAKNA Cancer Research Laboratory, Institute of Bioscience, Universiti Putra Malaysia, Serdang 43400, Selangor, Malaysia

6. Department of Pharmaceutical Technology, Kulliyyah of Pharmacy, International Islamic University Malaysia, Jalan Sultan Ahmad Shah, Kuantan 25200, Pahang, Malaysia

7. Basic & Applied Scientific Research Centre, Imam Abdulrahman Bin Faisal University, Dammam 31441, Saudi Arabia

8. Department of Biology, College of Science, Imam Abdulrahman Bin Faisal University, Dammam 31441, Saudi Arabia

9. Institute of Systems Biology, Universiti Kebangsaan Malaysia (UKM), Bangi 43600, Malaysia

10. Department of Food Technology, Faculty of Food Science, Wadi Alshatti University, Libya

11. Faculty of Pharmacy & Health Sciences, Universitas Abdurrab, Jalan Riau Ujung, Pekanbaru 28292, Riau, Indonesia

12. Laboratory of Natural Products, Institute of Bioscience, Universiti Putra Malaysia, UPM Serdang 43400, Selangor, Malaysia

13. Faculty of Industrial Sciences & Technology, Universiti Malaysia Pahang, Lebuhraya Tun Razak, Gambang 26300, Pahang, Malaysia

14. Drugs & Herbal Research Centre, Faculty of Pharmacy, Universiti Kebangsaan Malaysia, Jalan Raja Muda Abdul Aziz, Kuala Lumpur 50300, Malaysia

Funder

Ministry of Higher Education (MOHE) Malaysia

Publisher

Informa UK Limited

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