Synthesis, in vitro screening and molecular docking of isoquinolinium-5-carbaldoximes as acetylcholinesterase and butyrylcholinesterase reactivators-Reference-Cited by-同舟云学术

Synthesis, in vitro screening and molecular docking of isoquinolinium-5-carbaldoximes as acetylcholinesterase and butyrylcholinesterase reactivators

Published:2020-01-01 Issue:1 Volume:35 Page:478-488
ISSN:1475-6366
Container-title:Journal of Enzyme Inhibition and Medicinal Chemistry
language:en
Short-container-title:Journal of Enzyme Inhibition and Medicinal Chemistry

Author:

Malinak David¹²^ORCID,Dolezal Rafael¹²^ORCID,Hepnarova Vendula²³^ORCID,Hozova Miroslava²,Andrys Rudolf¹^ORCID,Bzonek Petr¹³,Racakova Veronika⁴,Korabecny Jan²³^ORCID,Gorecki Lukas²^ORCID,Mezeiova Eva²^ORCID,Psotka Miroslav¹²^ORCID,Jun Daniel²³^ORCID,Kuca Kamil¹²^ORCID,Musilek Kamil¹²^ORCID

Affiliation:

1. Department of Chemistry, Faculty of Science, University of Hradec Kralove, Hradec Kralove, Czech Republic

2. Biomedical Research Centre, University Hospital in Hradec Kralove, Hradec Kralove, Czech Republic

3. Department of Toxicology and Military Pharmacy, Faculty of Military Health Sciences, University of Defence, Hradec Kralove, Czech Republic

4. Faculty of Informatics and Management, Center for Basic and Applied Research, University of Hradec Kralove, Hradec Kralove, Czech Republic

Funder

Czech Science Foundation

Publisher

Informa UK Limited

Subject

Drug Discovery,Pharmacology,General Medicine

Link

https://www.tandfonline.com/doi/pdf/10.1080/14756366.2019.1710501

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2. Ligand-based 3D QSAR analysis of reactivation potency of mono- and bis-pyridinium aldoximes toward VX-inhibited rat acetylcholinesterase

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