The three-tails approach as a new strategy to improve selectivity of action of sulphonamide inhibitors against tumour-associated carbonic anhydrase IX and XII-Reference-Cited by-同舟云学术

The three-tails approach as a new strategy to improve selectivity of action of sulphonamide inhibitors against tumour-associated carbonic anhydrase IX and XII

Published:2022-03-21 Issue:1 Volume:37 Page:930-939
ISSN:1475-6366
Container-title:Journal of Enzyme Inhibition and Medicinal Chemistry
language:en
Short-container-title:Journal of Enzyme Inhibition and Medicinal Chemistry

Author:

Bonardi Alessandro¹²,Bua Silvia¹,Combs Jacob³,Lomelino Carrie³,Andring Jacob³,Osman Sameh Mohamed⁴,Toti Alessandra¹^ORCID,Di Cesare Mannelli Lorenzo¹^ORCID,Gratteri Paola²,Ghelardini Carla¹,McKenna Robert³,Nocentini Alessio¹^ORCID,Supuran Claudiu T.¹^ORCID

Affiliation:

1. Department NEUROFARBA – Pharmaceutical and Nutraceutical Section, University of Firenze, Florence, Italy

2. Department NEUROFARBA – Pharmaceutical and Nutraceutical Section, Laboratory of Molecular Modeling Cheminformatics & QSAR, University of Firenze, Florence, Italy

3. Department of Biochemistry and Molecular Biology, College of Medicine, University of Florida, Gainesville, FL, USA

4. Chemistry Department, College of Science, King Saud University, Riyadh, Saudi Arabia

Funder

Ministero dell'Istruzione, dell'Università e della Ricerca

Publisher

Informa UK Limited

Subject

Drug Discovery,Pharmacology,General Medicine

Link

https://www.tandfonline.com/doi/pdf/10.1080/14756366.2022.2053526

Reference59 articles.

1. Interfering with pH regulation in tumours as a therapeutic strategy