Triazoloquinoxalines-based DNA intercalators-Topo II inhibitors: design, synthesis, docking, ADMET and anti-proliferative evaluations-Reference-Cited by-同舟云学术

Triazoloquinoxalines-based DNA intercalators-Topo II inhibitors: design, synthesis, docking, ADMET and anti-proliferative evaluations

Published:2022-05-29 Issue:1 Volume:37 Page:1556-1567
ISSN:1475-6366
Container-title:Journal of Enzyme Inhibition and Medicinal Chemistry
language:en
Short-container-title:Journal of Enzyme Inhibition and Medicinal Chemistry

Author:

Elwan Alaa¹^ORCID,Sakr Helmy¹,El-Helby Abdel-Ghany A.¹,El-morsy Ahmed²,Abdelgawad Mohamed A.³^ORCID,Ghoneim Mohammed M.⁴^ORCID,El-Sherbiny Mohamed⁵⁶^ORCID,El-Adl Khaled¹⁷^ORCID

Affiliation:

1. Pharmaceutical Medicinal Chemistry & Drug Design Department, Faculty of Pharmacy (Boys), Al-Azhar University, Cairo, Egypt

2. Pharmaceutical Chemistry Department, College of Pharmacy, The Islamic University, Najaf, Iraq

3. Department of Pharmaceutical Chemistry, College of Pharmacy, Jouf University, Sakaka, Saudi Arabia

4. Department of Pharmacy Practice, Faculty of Pharmacy, AlMaarefa University, Ad Diriyah, Saudi Arabia

5. Department of Basic Medical Sciences, College of Medicine, AlMaarefa University, Riyadh, Saudi Arabia

6. Department of Anatomy, Faculty of Medicine, Mansoura University, Mansoura, Egypt

7. Chemistry Department, Faculty of Pharmacy, Heliopolis University for Sustainable Development, Cairo, Egypt

Funder

AlMaarefa University researchers supporting program

Publisher

Informa UK Limited

Subject

Drug Discovery,Pharmacology,General Medicine

Link

https://www.tandfonline.com/doi/pdf/10.1080/14756366.2022.2080205

Reference52 articles.

1. A DNA Intercalation Methodology for an Efficient Prediction of Ligand Binding Pose and Energetics

2. Intercalators as Anticancer Drugs

3. Intercalative Binding of Small Molecules to Nucleic Acids

4. Noncovalent interactions with DNA: An overview

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