Kinetic and thermodynamic characterisation of HIV-protease inhibitors against E35D↑G↑S mutant in the South African HIV-1 subtype C protease-Reference-Cited by-同舟云学术

Kinetic and thermodynamic characterisation of HIV-protease inhibitors against E35D↑G↑S mutant in the South African HIV-1 subtype C protease

Published:2019-01-01 Issue:1 Volume:34 Page:1451-1456
ISSN:1475-6366
Container-title:Journal of Enzyme Inhibition and Medicinal Chemistry
language:en
Short-container-title:Journal of Enzyme Inhibition and Medicinal Chemistry

Author:

Maseko Sibusiso¹^ORCID,Padayachee Eden¹,Maphumulo Siyabonga¹,Govender Thavendran¹,Sayed Yasien²,Maguire Glenn¹³,Lin Johnson⁴,Naicker Tricia¹,Baijnath Sooraj¹,Gerhardus Kruger Hendrik¹^ORCID

Affiliation:

1. Catalysis and Peptide Research Unit, School of Health Sciences, University of KwaZulu-Natal, Durban, South Africa;

2. Protein Structure-Function Research Unit, School of Molecular and Cell Biology, University of the Witwatersrand, Wits, South Africa;

3. School of Chemistry and Physics, University of KwaZulu-Natal, Durban, South Africa;

4. School of Life Sciences, University of KwaZulu-Natal, Durban, South Africa

Publisher

Informa UK Limited

Subject

Drug Discovery,Pharmacology,General Medicine

Link

https://www.tandfonline.com/doi/pdf/10.1080/14756366.2019.1636234

Reference25 articles.

1. Declining Morbidity and Mortality among Patients with Advanced Human Immunodeficiency Virus Infection

2. HIV-1 Antiretroviral Drug Therapy

3. Darunavir, a conceptually new HIV-1 protease inhibitor for the treatment of drug-resistant HIV

4. Molecular Basis for Drug Resistance in HIV-1 Protease

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