Synthesis, cyclooxygenase inhibition, anti-inflammatory evaluation and ulcerogenic liability of new 1,5-diarylpyrazole derivatives
Author:
Affiliation:
1. Department of Pharmaceutical Organic Chemistry, Beni-Suef University, Beni-Suef, Egypt,
2. Biochemistry Department, Cairo General Hospital, Cairo, Egypt, and
3. Pharmacology Department, Faculty of Veterinary, Cairo University, Cairo, Egypt
Publisher
Informa UK Limited
Subject
Drug Discovery,Pharmacology,General Medicine
Link
https://www.tandfonline.com/doi/pdf/10.1080/14756366.2016.1201815
Reference29 articles.
1. Inhibition of soluble epoxide hydrolase enhances the anti-inflammatory effects of aspirin and 5-lipoxygenase activation protein inhibitor in a murine model
2. COX-3, a cyclooxygenase-1 variant inhibited by acetaminophen and other analgesic/antipyretic drugs: Cloning, structure, and expression
3. Rationally Designed Multitarget Agents Against Inflammation and Pain
4. Selectivity of nonsteroidal antiinflammatory drugs as inhibitors of constitutive and inducible cyclooxygenase.
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