Comparative investigation of the in vitro inhibitory potencies of 13-epimeric estrones and D-secoestrones towards 17β-hydroxysteroid dehydrogenase type 1-Reference-Cited by-同舟云学术

Comparative investigation of the in vitro inhibitory potencies of 13-epimeric estrones and D-secoestrones towards 17β-hydroxysteroid dehydrogenase type 1

Published:2016-07-18 Issue:sup3 Volume:31 Page:61-69
ISSN:1475-6366
Container-title:Journal of Enzyme Inhibition and Medicinal Chemistry
language:en
Short-container-title:Journal of Enzyme Inhibition and Medicinal Chemistry

Author:

Herman Bianka Edina¹,Szabó Johanna²,Bacsa Ildikó²,Wölfling János²,Schneider Gyula²,Bálint Mónika³,Hetényi Csaba⁴,Mernyák Erzsébet²,Szécsi Mihály¹

Affiliation:

1. 1st Department of Medicine, University of Szeged, Szeged, Hungary,

2. Department of Organic Chemistry, University of Szeged, Szeged, Hungary,

3. Department of Biochemistry, Eötvös Loránd University, Budapest, Hungary, and

4. MTA-ELTE Molecular Biophysics Research Group, Hungarian Academy of Sciences, Budapest, Hungary

Publisher

Informa UK Limited

Subject

Drug Discovery,Pharmacology,General Medicine

Link

https://www.tandfonline.com/doi/pdf/10.1080/14756366.2016.1204610

Reference52 articles.

1. Integrated view on 17beta-hydroxysteroid dehydrogenases

2. 17β-Hydroxysteroid dehydrogenases (17β-HSDs) as therapeutic targets: Protein structures, functions, and recent progress in inhibitor development

3. Multifunctionality of human 17β-hydroxysteroid dehydrogenases

4. Characteristics of human types 1, 2 and 3 17β-hydroxysteroid dehydrogenase activities: Oxidation/reduction and inhibition

5. Human Estrogenic 17β-Hydroxysteroid Dehydrogenase: Predominance of Estrone Reduction and Its Induction by NADPH

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