Discovery of potent tubulin inhibitors targeting the colchicine binding site via structure-based lead optimization and antitumor evaluation-Reference-Cited by-同舟云学术

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Discovery of potent tubulin inhibitors targeting the colchicine binding site via structure-based lead optimization and antitumor evaluation

Published:2023-01-11 Issue:1 Volume:38 Page:
ISSN:1475-6366
Container-title:Journal of Enzyme Inhibition and Medicinal Chemistry
language:en
Short-container-title:Journal of Enzyme Inhibition and Medicinal Chemistry

Author:

Liu Wei¹,He Youyou¹²,Guo Zhongjie²,Wang Miaomiao¹,Han Xiaodong²,Jia Hairui¹,He Jin²,Miao Shanshan²,Wang Shengzheng²

Affiliation:

1. Faculty of Pharmacy, School of Food and Biological Engineering, Shaanxi University of Science and Technology, Xi’an, China

2. Department of Medicinal Chemistry and Pharmaceutical Analysis, School of Pharmacy, Fourth Military Medical University, Xi’an, China

Funder

Natural Science Basic Research Plan in Shaanxi Province

Publisher

Informa UK Limited

Subject

Drug Discovery,Pharmacology,General Medicine

Link

https://www.tandfonline.com/doi/pdf/10.1080/14756366.2022.2155815

Reference43 articles.

1. Structure-Guided Design, Synthesis, and Biological Evaluation of (2-(1H-Indol-3-yl)-1H-imidazol-4-yl)(3,4,5-trimethoxyphenyl) Methanone (ABI-231) Analogues Targeting the Colchicine Binding Site in Tubulin

2. Microtubules as a target for anticancer drugs

3. Drugs that target dynamic microtubules: A new molecular perspective

4. Tubulin structure: insights into microtubule properties and functions

5. Structural Optimization of Indole Derivatives Acting at Colchicine Binding Site as Potential Anticancer Agents

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1. Discovery of novel amide derivatives against VEGFR-2/tubulin with potent antitumor and antiangiogenic activity;Bioorganic Chemistry;2024-10

2. Tubulin inhibitors. Selected scaffolds and main trends in the design of novel anticancer and antiparasitic agents;Bioorganic Chemistry;2024-02

3. Recognition of arylmethylidene derivatives of imidazothiazolotriazinones as novel tubulin polymerization inhibitors;RSC Medicinal Chemistry;2024

4. Design, synthesis and antiproliferative evaluation of lipidated 1,3-diaryl propenones and their cyclized pyrimidine derivatives as tubulin polymerization inhibitors;Results in Chemistry;2023-12

5. Discovery of Platinum^IV–Artesunate Multiaction Prodrugs as Potent Antitumor and Antimalarial Agents;Journal of Medicinal Chemistry;2023-06-12

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