Tetralone derivatives are MIF tautomerase inhibitors and attenuate macrophage activation and amplify the hypothermic response in endotoxemic mice-Reference-Cited by-同舟云学术

Tetralone derivatives are MIF tautomerase inhibitors and attenuate macrophage activation and amplify the hypothermic response in endotoxemic mice

Published:2021-01-01 Issue:1 Volume:36 Page:1356-1368
ISSN:1475-6366
Container-title:Journal of Enzyme Inhibition and Medicinal Chemistry
language:en
Short-container-title:Journal of Enzyme Inhibition and Medicinal Chemistry

Author:

Garai János¹^ORCID,Krekó Marcell²^ORCID,Őrfi László²^ORCID,Jakus Péter Balázs³^ORCID,Rumbus Zoltán⁴^ORCID,Kéringer Patrik⁴^ORCID,Garami András⁴^ORCID,Vámos Eszter³^ORCID,Kovács Dominika³^ORCID,Bagóné Vántus Viola³^ORCID,Radnai Balázs³^ORCID,Lóránd Tamás³^ORCID

Affiliation:

1. Department of Pathophysiology, Institute for Translational Medicine, University of Pécs, Medical School, Pécs, Hungary

2. Department of Pharmaceutical Chemistry, Semmelweis University, Budapest, Hungary

3. Department of Biochemistry and Medical Chemistry, University of Pécs, Medical School, Pécs, Hungary

4. Department of Thermophysiology, Institute for Translational Medicine, University of Pécs, Medical School, Pécs, Hungary

Funder

János Bolyai Research Scholarship of the Hungarian Academy of Sciences

National Research, Development and Innovation Office

Medical School, University of Pecs

Higher Education Institutional Excellence Program of the Ministry of Human Capacities in Hungary

European Union, co-financed by the European Social Fund

Ministry of Finance, Hungary

Publisher

Informa UK Limited

Subject

Drug Discovery,Pharmacology,General Medicine

Link

https://www.tandfonline.com/doi/pdf/10.1080/14756366.2021.1916010

Reference90 articles.

1. Mechanism of a Reaction in Vitro Associated with Delayed-Type Hypersensitivity

2. Delayed hypersensitivity in vitro: its mediation by cell-free substances formed by lymphoid cell-antigen interaction.

3. The MIF Handbook

4. Macrophage Migration Inhibitory Factor: A Probable Link between Inflammation and Cancer

5. Crystallization and Preliminary X-Ray Analysis of Humand-Dopachrome Tautomerase

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