Targeting allosteric sites of human aromatase: a comprehensive in-silico and in-vitro workflow to find potential plant-based anti-breast cancer therapeutics-Reference-Cited by-同舟云学术

Targeting allosteric sites of human aromatase: a comprehensive in-silico and in-vitro workflow to find potential plant-based anti-breast cancer therapeutics

Published:2021-01-01 Issue:1 Volume:36 Page:1333-1344
ISSN:1475-6366
Container-title:Journal of Enzyme Inhibition and Medicinal Chemistry
language:en
Short-container-title:Journal of Enzyme Inhibition and Medicinal Chemistry

Author:

Alhadrami Hani A.¹²³,Sayed Ahmed M.⁴,Melebari Sami A.³,Khogeer Asem A.⁵,Abdulaal Wesam H.⁶,Al-Fageeh Mohamed B.⁷,Algahtani Mohammad⁸,Rateb Mostafa E.⁹

Affiliation:

1. Department of Medical Laboratory Technology, Faculty of Applied Medical Sciences, King Abdulaziz University, Jeddah, Saudi Arabia

2. Molecular Diagnostic Lab, King Abdulaziz University Hospital, King Abdulaziz University, Jeddah, Saudi Arabia

3. Molecular Diagnostic Unit, The Regional Laboratory in Makkah, Ministry of Health, Makkah, Kingdom of Saudi Arabia

4. Department of Pharmacognosy, Faculty of Pharmacy, Nahda University, Beni Suef, Egypt

5. Plan and Research Department, General Directorate of Health Affairs, Makkah region, Ministry of Health, Makkah, Kingdom of Saudi Arabia

6. Department of Biochemistry, Faculty of Science, King Abdulaziz University, Jeddah, Saudi Arabia

7. General Directorate for Funds and Grants (GDFG), King Abdulaziz City for Science and Technology, Riyadh, Saudi Arabia

8. Department of Laboratory and Blood Bank, Security Forces Hospital Program, Mecca, Saudi Arabia

9. School of Computing, Engineering & Physical Sciences, University of the West of Scotland, Paisley, UK

Funder

Deanship of Scientific Research (DSR), King Abdulaziz University, Jeddah

Publisher

Informa UK Limited

Subject

Drug Discovery,Pharmacology,General Medicine

Link

https://www.tandfonline.com/doi/pdf/10.1080/14756366.2021.1937145

Reference48 articles.

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3. Selective estrogen receptor modulators (SERMs): Mechanisms of anticarcinogenesis and drug resistance

4. Recent Progress in the Discovery of Next Generation Inhibitors of Aromatase from the Structure–Function Perspective

5. Acquired resistance to aromatase inhibitors: where we stand!

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