Design, synthesis, docking, MD simulations, and anti-proliferative evaluation of thieno[2,3- <i>d</i> ]pyrimidine derivatives as new EGFR inhibitors-Reference-Cited by-同舟云学术

Design, synthesis, docking, MD simulations, and anti-proliferative evaluation of thieno[2,3- d ]pyrimidine derivatives as new EGFR inhibitors

Published:2023-06-08 Issue:1 Volume:38 Page:
ISSN:1475-6366
Container-title:Journal of Enzyme Inhibition and Medicinal Chemistry
language:en
Short-container-title:Journal of Enzyme Inhibition and Medicinal Chemistry

Author:

Sobh Eman A.¹,Dahab Mohammed A.²^ORCID,Elkaeed Eslam B.³,Alsfouk Aisha A.⁴,Ibrahim Ibrahim M.⁵,Metwaly Ahmed M.⁶⁷^ORCID,Eissa Ibrahim H.²^ORCID

Affiliation:

1. Department of Pharmaceutical Chemistry, Faculty of Pharmacy, Menoufia University, Menoufia, Egypt

2. Pharmaceutical Medicinal Chemistry & Drug Design Department, Faculty of Pharmacy (Boys), Al-Azhar University, Cairo, Egypt

3. Department of Pharmaceutical Sciences, College of Pharmacy, AlMaarefa University, Riyadh, Saudi Arabia

4. Department of Pharmaceutical Sciences, College of Pharmacy, Princess Nourah bint Abdulrahman University, Riyadh, Saudi Arabia

5. Biophysics Department, Faculty of Science, Cairo University, Cairo, Egypt

6. Pharmacognosy and Medicinal Plants Department, Faculty of Pharmacy (Boys), Al-Azhar University, Cairo, Egypt

7. Biopharmaceutical Products Research Department, Genetic Engineering and Biotechnology Research Institute, City of Scientific Research and Technological Applications (SRTA-City), Alexandria, Egypt

Funder

AlMaarefa University

Princess Nourah bint Abdulrahman University

Publisher

Informa UK Limited

Subject

Drug Discovery,Pharmacology,General Medicine

Link

https://www.tandfonline.com/doi/pdf/10.1080/14756366.2023.2220579

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