Mixed and non-competitive enzyme inhibition: underlying mechanisms and mechanistic irrelevance of the formal two-site model-Reference-Cited by-同舟云学术

Mixed and non-competitive enzyme inhibition: underlying mechanisms and mechanistic irrelevance of the formal two-site model

Published:2023-08-14 Issue:1 Volume:38 Page:
ISSN:1475-6366
Container-title:Journal of Enzyme Inhibition and Medicinal Chemistry
language:en
Short-container-title:Journal of Enzyme Inhibition and Medicinal Chemistry

Author:

Pesaresi Alessandro¹

Affiliation:

1. Istituto di Cristallografia – Consiglio Nazionale delle Ricerche, Trieste, Italy

Publisher

Informa UK Limited

Subject

Drug Discovery,Pharmacology,General Medicine

Link

https://www.tandfonline.com/doi/pdf/10.1080/14756366.2023.2245168

Reference63 articles.

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3. Evaluation of Enzyme Inhibitors in Drug Discovery

4. Novel Antimycobacterial Compounds Suppress NAD Biogenesis by Targeting a Unique Pocket of NaMN Adenylyltransferase

5. Copeland RA, Anderson PS. Enzymes and Enzyme Inhibitors” in Textbook of Drug Design and Discovery. 3rd ed., P. Krogsgaard-Larsen, T. Liljefors, U. Madsen, editors. New York: Taylor and Francis; 2002

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