Synthesis and structure–activity relationships of 2- and/or 4-halogenated 13β- and 13α-estrone derivatives as enzyme inhibitors of estrogen biosynthesis-Reference-Cited by-同舟云学术

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Synthesis and structure–activity relationships of 2- and/or 4-halogenated 13β- and 13α-estrone derivatives as enzyme inhibitors of estrogen biosynthesis

Published:2018-01-01 Issue:1 Volume:33 Page:1271-1282
ISSN:1475-6366
Container-title:Journal of Enzyme Inhibition and Medicinal Chemistry
language:en
Short-container-title:Journal of Enzyme Inhibition and Medicinal Chemistry

Author:

Bacsa Ildikó¹,Herman Bianka Edina²,Jójárt Rebeka¹,Herman Kevin Stefán¹,Wölfling János¹,Schneider Gyula¹,Varga Mónika³,Tömböly Csaba⁴,Rižner Tea Lanišnik⁵,Szécsi Mihály²,Mernyák Erzsébet¹

Affiliation:

1. Department of Organic Chemistry, University of Szeged, Szeged, Hungary;

2. 1st Department of Medicine, University of Szeged, Szeged, Hungary;

3. Department of Microbiology, University of Szeged, University of Szeged, Szeged, Hungary;

4. Laboratory of Chemical Biology, Institute of Biochemistry, Biological Research Centre of the Hungarian Academy of Sciences, Szeged, Hungary

5. Institute of Biochemistry, Faculty of Medicine, University of Ljubljana, Ljubljana, Slovenia

Funder

Hungarian Academy of Sciences

Ministry Of Human Capacities

Publisher

Informa UK Limited

Subject

Drug Discovery,Pharmacology,General Medicine

Link

https://www.tandfonline.com/doi/pdf/10.1080/14756366.2018.1490731

Reference39 articles.

1. The Molecular Biology, Biochemistry, and Physiology of Human Steroidogenesis and Its Disorders

2. Substrate-Dependent Inhibition of Organic Anion Transporting Polypeptide 1B1: Comparative Analysis with Prototypical Probe Substrates Estradiol-17β-Glucuronide, Estrone-3-Sulfate, and Sulfobromophthalein

3. Estrogen O-sulfamates and their analogues: Clinical steroid sulfatase inhibitors with broad potential

4. Aromatase, estrone sulfatase, and 17β-hydroxysteroid dehydrogenase: Structure–function studies and inhibitor development

5. Structure–activity relationships of 2-, 4-, or 6-substituted estrogens as aromatase inhibitors

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1. Cytotoxic effect of 13α-estrane derivatives on breast, endometrial and ovarian cancer cell lines;The Journal of Steroid Biochemistry and Molecular Biology;2023-09

2. Synthesis and Antiproliferative Activity of Steroidal Diaryl Ethers;Molecules;2023-01-25

3. Inhibitor of Glucosinolate Sulfatases as a Potential Friendly Insecticide to Control Plutella xylostella;Journal of Agricultural and Food Chemistry;2022-10-17

4. Dual Targeting of Steroid Sulfatase and 17β-Hydroxysteroid Dehydrogenase Type 1 by a Novel Drug-Prodrug Approach: A Potential Therapeutic Option for the Treatment of Endometriosis;Journal of Medicinal Chemistry;2022-08-22

5. Selective antiproliferative effect of C-2 halogenated 13α-estrones on cells expressing Organic anion-transporting polypeptide 2B1 (OATP2B1);Toxicology and Applied Pharmacology;2021-10

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