Inhibition studies on a panel of human carbonic anhydrases with N1-substituted secondary sulfonamides incorporating thiazolinone or imidazolone-indole tails-Reference-Cited by-同舟云学术

Inhibition studies on a panel of human carbonic anhydrases with N1-substituted secondary sulfonamides incorporating thiazolinone or imidazolone-indole tails

Published:2018-01-01 Issue:1 Volume:33 Page:629-638
ISSN:1475-6366
Container-title:Journal of Enzyme Inhibition and Medicinal Chemistry
language:en
Short-container-title:Journal of Enzyme Inhibition and Medicinal Chemistry

Author:

Awadallah Fadi M.¹,Bua Silvia²,Mahmoud Walaa R.¹,Nada Hossam H.³,Nocentini Alessio²,Supuran Claudiu T.²

Affiliation:

1. Pharmaceutical Chemistry Department, Faculty of Pharmacy, Cairo University, Cairo, Egypt;

2. Department NEUROFARBA – Pharmaceutical and Nutraceutical Section, University of Firenze, Firenze, Italy;

3. Pharmaceutical Chemistry Department, Faculty of Pharmacy, Badr University, Cairo, Egypt

Funder

University of Florence

Publisher

Informa UK Limited

Subject

Drug Discovery,Pharmacology,General Medicine

Link

https://www.tandfonline.com/doi/pdf/10.1080/14756366.2018.1446432

Reference40 articles.

1. Carbon- versus sulphur-based zinc binding groups for carbonic anhydrase inhibitors?

2. Carbonic anhydrases: novel therapeutic applications for inhibitors and activators

3. Multiple Binding Modes of Inhibitors to Carbonic Anhydrases: How to Design Specific Drugs Targeting 15 Different Isoforms?

4. Drug Design of Zinc-Enzyme Inhibitors

5. Combining the tail and the ring approaches for obtaining potent and isoform-selective carbonic anhydrase inhibitors: Solution and X-ray crystallographic studies

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