Design, synthesis, and in vitro evaluation of BP-1-102 analogs with modified hydrophobic fragments for STAT3 inhibition-Reference-Cited by-同舟云学术

Design, synthesis, and in vitro evaluation of BP-1-102 analogs with modified hydrophobic fragments for STAT3 inhibition

Published:2021-01-01 Issue:1 Volume:36 Page:410-424
ISSN:1475-6366
Container-title:Journal of Enzyme Inhibition and Medicinal Chemistry
language:en
Short-container-title:Journal of Enzyme Inhibition and Medicinal Chemistry

Author:

Oleksak Patrik¹,Psotka Miroslav¹^ORCID,Vancurova Marketa²,Sapega Olena³,Bieblova Jana³,Reinis Milan³^ORCID,Rysanek David²,Mikyskova Romana³,Chalupova Katarina¹^ORCID,Malinak David¹^ORCID,Svobodova Jana¹^ORCID,Andrys Rudolf¹^ORCID,Rehulkova Helena¹^ORCID,Skopek Vojtech¹,Ngoc Lam Pham¹,Bartek Jiri²⁴,Hodny Zdenek²^ORCID,Musilek Kamil¹^ORCID

Affiliation:

1. Department of Chemistry, Faculty of Science, University of Hradec Kralove, Hradec Kralove, Czech Republic

2. Department of Genome Integrity, Institute of Molecular Genetics of the Czech Academy of Sciences, Prague, Czech Republic

3. Laboratory of Immunological and Tumour Models, Institute of Molecular Genetics of the Czech Academy of Sciences, Prague, Czech Republic

4. Genome Integrity Unit, Danish Cancer Society Research Center, Copenhagen, Denmark

Funder

Czech Science Foundation

Institutional Grant

University of Hradec Kralove

Publisher

Informa UK Limited

Subject

Drug Discovery,Pharmacology,General Medicine

Link

https://www.tandfonline.com/doi/pdf/10.1080/14756366.2020.1871336

Reference39 articles.

1. Canonical and non-canonical JAK/STAT transcriptional targets may be involved in distinct and overlapping cellular processes

2. STATs and Gene Regulation

3. The role of STATs in transcriptional control and their impact on cellular function

4. The STATs of cancer — new molecular targets come of age

5. Stat3 as an Oncogene

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