New classes of potent heparanase inhibitors from ligand-based virtual screening-Reference-Cited by-同舟云学术

New classes of potent heparanase inhibitors from ligand-based virtual screening

Published:2020-01-01 Issue:1 Volume:35 Page:1685-1696
ISSN:1475-6366
Container-title:Journal of Enzyme Inhibition and Medicinal Chemistry
language:en
Short-container-title:Journal of Enzyme Inhibition and Medicinal Chemistry

Author:

Pala Daniele¹^ORCID,Scalvini Laura¹^ORCID,Elisi Gian Marco¹^ORCID,Lodola Alessio¹^ORCID,Mor Marco¹^ORCID,Spadoni Gilberto²^ORCID,Ferrara Fabiana F.³,Pavoni Emiliano³,Roscilli Giuseppe³,Milazzo Ferdinando M.⁴,Battistuzzi Gianfranco⁴,Rivara Silvia¹^ORCID,Giannini Giuseppe⁴^ORCID

Affiliation:

1. Dipartimento di Scienze degli Alimenti e del Farmaco, Università degli Studi di Parma, Parma, Italy

2. Dipartimento di Scienze Biomolecolari, Università degli Studi di Urbino “Carlo Bo”, Urbino, Italy

3. Takis s.r.l., Roma, Italy

4. R&D Alfasigma S.p.A., Roma, Italy

Funder

Leadiant Biosciences S.A.

Publisher

Informa UK Limited

Subject

Drug Discovery,Pharmacology,General Medicine

Link

https://www.tandfonline.com/doi/pdf/10.1080/14756366.2020.1811701

Reference56 articles.

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4. Heparanase: a rainbow pharmacological target associated to multiple pathologies including rare diseases

5. The Functions of Heparanase in Human Diseases

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