10β-Hydroxyestra-1,4-diene-3,17-dione as potential antiproliferative agent: in vitro biological evaluation and in silico studies-Reference-Cited by-同舟云学术

10β-Hydroxyestra-1,4-diene-3,17-dione as potential antiproliferative agent: in vitro biological evaluation and in silico studies

Published:2022-02-15 Issue:24 Volume:36 Page:6459-6463
ISSN:1478-6419
Container-title:Natural Product Research
language:en
Short-container-title:Natural Product Research

Author:

Canário Catarina¹,Matias Mariana¹,Brito Vanessa de¹,Cruz-Vicente Pedro¹²,Soeiro Pedro¹,Santos Adriana O.¹,Falcão Amílcar³⁴⁵,Silvestre Samuel¹³,Alves Gilberto¹

Affiliation:

1. CICS-UBI – Health Sciences Research Centre, University of Beira Interior, Covilhã, Portugal

2. UCIBIO – Applied Molecular Biosciences Unit, Chemistry Department, Sciences and Technology Faculty, Nova Lisbon University, Costa da Caparica, Portugal

3. CNC – Center for Neuroscience and Cell Biology, University of Coimbra, Coimbra, Portugal

4. Laboratory of Pharmacology, Faculty of Pharmacy, University of Coimbra, Coimbra, Portugal

5. CIBIT - Coimbra Institute for Biomedical Imaging and Translational Research, University of Coimbra, Coimbra, Portugal

Funder

Funda??o para a Ci?ncia e a Tecnologia

FEDER funds through the POCI - COMPETE 2020 - Operational Program Competitiveness and Internationalization in Axis I - Strengthening research, technological development and innovation

Publisher

Informa UK Limited

Subject

Organic Chemistry,Plant Science,Biochemistry,Analytical Chemistry

Link

https://www.tandfonline.com/doi/pdf/10.1080/14786419.2022.2039136

Reference12 articles.

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3. Molecular Interactions between Estrogen Receptor and Its Ligand Studied by the ab Initio Fragment Molecular Orbital Method

4. Aromatase, estrone sulfatase, and 17β-hydroxysteroid dehydrogenase: Structure–function studies and inhibitor development

5. Practical one-pot conversion of 17β-estradiol to 10β-hydroxy- (p-quinol) and 10β-chloro-17β-hydroxyestra-1,4-dien-3-one