Design of new CD38 inhibitors based on CoMFA modelling and molecular docking analysis of 4‑amino-8-quinoline carboxamides and 2,4-diamino-8-quinazoline carboxamides
Author:
Affiliation:
1. Department of Chemistry, Faculty of Science, University of Kurdistan, Sanandaj, Iran
Publisher
Informa UK Limited
Subject
Drug Discovery,Molecular Medicine,General Medicine,Bioengineering
Link
https://www.tandfonline.com/doi/pdf/10.1080/1062936X.2018.1545695
Reference50 articles.
1. CD38-targeting antibodies in multiple myeloma: mechanisms of action and clinical experience
2. The CD38 Lymphocyte Differentiation Marker: New Insight into Its Ectoenzymatic Activity and Its Role as a Signal Transducer
3. Crystal Structure of Human CD38 Extracellular Domain
4. CD38 at the junction between prognostic marker and therapeutic target
5. The metamorphosis of a molecule: from soluble enzyme to the leukocyte receptor CD38
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