Novel Procedure for the Coupling of Sterically Hindered Electron-Deficient Anilines to the 6-Position of the Purine Core-Reference-Cited by-同舟云学术

Novel Procedure for the Coupling of Sterically Hindered Electron-Deficient Anilines to the 6-Position of the Purine Core

Published:2011-07-27 Issue:21 Volume:41 Page:3246-3250
ISSN:0039-7911
Container-title:Synthetic Communications
language:en
Short-container-title:Synthetic Communications

Author:

Leenders Ruben¹,Heeres Jan²,Vandenput Dirk¹,Guillemont Jérôme³,Lewi Paul²

Affiliation:

1. a Mercachem BV , Nijmegen , the Netherlands

2. b Janssen Research Foundation, Center for Molecular Design , Vosselaar , Belgium

3. c Johnson and Johnson Pharmaceutical Research and Development, Medicinal Chemistry Department , Val de Reuil , France

Publisher

Informa UK Limited

Subject

Organic Chemistry

Link

https://www.tandfonline.com/doi/pdf/10.1080/00397911.2010.517615

Reference10 articles.

1. A novel route to 2,4-dianilino-substituted pyrimidines

2. Janssen , P. Lewi , P. de Jonge , M. Koymans , L. Daeyaert , F. Heeres , J. Vinkers , H. Leenders , R. Vandenput , D. HIV replication inhibiting purine derivatives . WO Patent 2005/028479, 2005 .

3. 9-Benzyl-6-(dimethylamino)-9H-purines with antirhinovirus activity

4. Antirhinovirus activity of 6-anilino-9-benzyl-2-chloro-9H-purines

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