Design, synthesis and biological evaluation of some 2-(6-nitrobenzo[d]thiazol-2-ylthio)-N-benzyl-N-(6-nitrobenzo[d]thiazol-2-yl)acetamide derivatives as selective DprE1 inhibitors-Reference-Cited by-同舟云学术

Design, synthesis and biological evaluation of some 2-(6-nitrobenzo[d]thiazol-2-ylthio)-N-benzyl-N-(6-nitrobenzo[d]thiazol-2-yl)acetamide derivatives as selective DprE1 inhibitors

Published:2019-08-01 Issue:20 Volume:49 Page:2696-2708
ISSN:0039-7911
Container-title:Synthetic Communications
language:en
Short-container-title:Synthetic Communications

Author:

Gawad Jineetkumar¹^ORCID,Bonde Chandrakant¹

Affiliation:

1. Department of Pharmaceutical Chemistry, School of Pharmacy and Technology Management, SVKM's NMIMS, Dhule, India

Publisher

Informa UK Limited

Subject

Organic Chemistry

Link

https://www.tandfonline.com/doi/pdf/10.1080/00397911.2019.1639756

Reference41 articles.

1. Design, Syntheses, and Anti-TB Activity of 1,3-Benzothiazinone Azide and Click Chemistry Products Inspired by BTZ043

2. Comparative Studies Evaluating Mouse Models Used for Efficacy Testing of Experimental Drugs against Mycobacterium tuberculosis

3. The DprE1 enzyme, one of the most vulnerable targets of Mycobacterium tuberculosis

4. Benzothiazinones Kill Mycobacterium tuberculosis by Blocking Arabinan Synthesis

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