Synthesis, biological activity, molecular docking studies of a novel series of 3-Aryl-7H-thiazolo[3,2-b]-1,2,4-triazin-7-one derivatives as the acetylcholinesterase inhibitors
Author:
Affiliation:
1. Key Laboratory of Structure-based Drug Design & Discovery, Ministry of Education, Shenyang Pharmaceutical University, Shenyang, China
2. School of Biomedical Sciences, Faculty of Medicine, The Chinese University of Hong Kong, Hong Kong SAR, China
Funder
National Natural Science Foundation of China
National Science Foundation of China
Program for Innovative Research Team of the Ministry of Education of China
Natural Science Foundation of Liaoning Province, China
Scientific Research Foundation of Department of Education of Liaoning Province
Publisher
Informa UK Limited
Subject
Molecular Biology,General Medicine,Structural Biology
Link
https://www.tandfonline.com/doi/pdf/10.1080/07391102.2020.1753576
Reference48 articles.
1. Key Challenges and Opportunities Associated with the Use of In Vitro Models to Detect Human DILI: Integrated Risk Assessment and Mitigation Plans
2. Structural Evidence That Human Acetylcholinesterase Inhibited by Tabun Ages through O-Dealkylation
3. Structures of Human Acetylcholinesterase in Complex with Pharmacologically Important Ligands
4. Molecular modeling studies on the interactions of aflatoxin B1 and its metabolites with the peripheral anionic site of human acetylcholinesterase
5. Acetylcholinesterase: From 3D structure to function
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