Synthesis, biological activity, molecular docking studies of a novel series of 3-Aryl-7H-thiazolo[3,2-b]-1,2,4-triazin-7-one derivatives as the acetylcholinesterase inhibitors-Reference-Cited by-同舟云学术

Synthesis, biological activity, molecular docking studies of a novel series of 3-Aryl-7H-thiazolo[3,2-b]-1,2,4-triazin-7-one derivatives as the acetylcholinesterase inhibitors

Published:2020-04-16 Issue:7 Volume:39 Page:2478-2489
ISSN:0739-1102
Container-title:Journal of Biomolecular Structure and Dynamics
language:en
Short-container-title:Journal of Biomolecular Structure and Dynamics

Author:

Jin Zhe¹,Zhang Chao¹,Liu Miao¹,Jiao Simeng¹,Zhao Jing¹,Liu Xiaoping¹,Lin Huangquan²,Chi-cheong Wan David²,Hu Chun¹

Affiliation:

1. Key Laboratory of Structure-based Drug Design & Discovery, Ministry of Education, Shenyang Pharmaceutical University, Shenyang, China

2. School of Biomedical Sciences, Faculty of Medicine, The Chinese University of Hong Kong, Hong Kong SAR, China

Funder

National Natural Science Foundation of China

National Science Foundation of China

Program for Innovative Research Team of the Ministry of Education of China

Natural Science Foundation of Liaoning Province, China

Scientific Research Foundation of Department of Education of Liaoning Province

Publisher

Informa UK Limited

Subject

Molecular Biology,General Medicine,Structural Biology

Link

https://www.tandfonline.com/doi/pdf/10.1080/07391102.2020.1753576

Reference48 articles.

1. Key Challenges and Opportunities Associated with the Use of In Vitro Models to Detect Human DILI: Integrated Risk Assessment and Mitigation Plans

2. Structural Evidence That Human Acetylcholinesterase Inhibited by Tabun Ages through O-Dealkylation

3. Structures of Human Acetylcholinesterase in Complex with Pharmacologically Important Ligands

4. Molecular modeling studies on the interactions of aflatoxin B1 and its metabolites with the peripheral anionic site of human acetylcholinesterase

5. Acetylcholinesterase: From 3D structure to function

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