Disposition and metabolism of [14C]-galunisertib, a TGF-βRI kinase/ALK5 inhibitor, following oral administration in healthy subjects and mechanistic prediction of the effect of itraconazole on galunisertib pharmacokinetics-Reference-Cited by-同舟云学术

Disposition and metabolism of [14C]-galunisertib, a TGF-βRI kinase/ALK5 inhibitor, following oral administration in healthy subjects and mechanistic prediction of the effect of itraconazole on galunisertib pharmacokinetics

Published:2017-05-16 Issue:4 Volume:48 Page:382-399
ISSN:0049-8254
Container-title:Xenobiotica
language:en
Short-container-title:Xenobiotica

Author:

Cassidy Kenneth C.¹,Gueorguieva Ivelina²,Miles Colin²,Rehmel Jessica¹,Yi Ping¹,Ehlhardt William J.¹

Affiliation:

1. Eli Lilly and Company, Lilly Corporate Center, Indianapolis, IN, USA and

2. Eli Lilly and Company Erl Wood, Windlesham, UK

Publisher

Informa UK Limited

Subject

Health, Toxicology and Mutagenesis,Pharmacology,Toxicology,Biochemistry,General Medicine

Link

https://www.tandfonline.com/doi/pdf/10.1080/00498254.2017.1323137

Reference27 articles.

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