1. Pfizer Worldwide Research and Development, La Jolla Laboratories, San Diego, CA, USA,
2. Department of Medicine, University of California San Diego, La Jolla, CA, USA,
3. Pfizer Worldwide Research and Development, Groton, CT, USA,
4. ORIC Pharmaceuticals, South San Francisco, CA, USA, and
5. Department of Pathology, University of California San Diego, La Jolla, CA, USA