The influence of temperature on the metabolic activity of CYP2C9, CYP2C19, and CYP3A4 genetic variants in vitro

Author:

Kojima Michiaki1,Machida Kanami1,Cho Sumie1,Watanabe Daichi2,Seki Hiroyuki2,Shimoji Miyuki3,Imaoka Ayuko1,Yamazaki Hiroshi4ORCID,Guengerich F. Peter5,Nakamura Katsunori3,Yamamoto Koujirou6,Akiyoshi Takeshi127,Ohtani Hisakazu1278

Affiliation:

1. Division of Clinical Pharmacokinetics, Faculty of Pharmacy, Keio University, Tokyo, Japan

2. Division of Clinical Pharmacokinetics, Graduate School of Pharmaceutical Sciences, Keio University, Tokyo, Japan

3. Department of Pharmacy, University of the Ryukyus Hospital, Okinawa, Japan

4. Laboratory of Drug Metabolism and Pharmacokinetics, Showa Pharmaceutical University, Tokyo, Machida, Japan

5. Department of Biochemistry, Vanderbilt University School of Medicine, Nashville, USA

6. Gunma University Graduate School of Medicine, Gunma, Japan

7. Division of Clinical Pharmacokinetics, School of Medicine, Keio University, Tokyo, Shinjuku, Japan

8. Department of Pharmacy, Keio University Hospital, Tokyo, Shinjuku, Japan

Funder

Japan Research Foundation for JSPS Kakenhi

United States National Institutes of Health

Publisher

Informa UK Limited

Subject

Health, Toxicology and Mutagenesis,Pharmacology,Toxicology,Biochemistry,General Medicine

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