Synthesis of S-mono- and S,O-bis-1,2,3-triazole linked 1,5-benzodiazepine conjugates and evaluation of their cytotoxic, anti-tyrosinase, and anti-cholinesterase activities-Reference-Cited by-同舟云学术

Synthesis of S-mono- and S,O-bis-1,2,3-triazole linked 1,5-benzodiazepine conjugates and evaluation of their cytotoxic, anti-tyrosinase, and anti-cholinesterase activities

Published:2017-03-21 Issue:7 Volume:192 Page:835-844
ISSN:1042-6507
Container-title:Phosphorus, Sulfur, and Silicon and the Related Elements
language:en
Short-container-title:Phosphorus, Sulfur, and Silicon and the Related Elements

Author:

Abdallah Wejdane¹²,Znati Mansour²,Regazzetti Anne³,Dargère Delphine³,Laprévote Olivier³,Ben Jannet Hichem²,Gharbi Rafik¹

Affiliation:

1. Laboratory of Applied Chemistry and Environment, Faculty of Science of Monastir, University of Monastir, Monastir, Tunisia

2. Laboratory of Heterocyclic Chemistry, Natural Products and Reactivity (LR11SE39), Team: Medicinal Chemistry and Natural Products and Reactivity, Faculty of Science of Monastir, University of Monastir, Monastir, Tunisia

3. Laboratory C-TAC Faculty of Pharmaceutical and Biological Sciences, Paris, France

Publisher

Informa UK Limited

Subject

Inorganic Chemistry,Organic Chemistry,Biochemistry

Link

https://www.tandfonline.com/doi/pdf/10.1080/10426507.2017.1287704

Reference49 articles.

1. Synthesis of 1,5-Benzodiazepine Derivatives Containing 1,2,3-Triazole Moiety via 1,3-Dipolar Cycloaddition Reaction

2. 1,5-Benzodiazepine derivatives as potential antimicrobial agents: design, synthesis, biological evaluation, and structure–activity relationships

3. 1,4-Benzodiazepines. Chemistry and Some Aspects of the Structure-Activity Relationship

4. New potent inhibitors of tyrosinase: Novel clues to binding of 1,3,4-thiadiazole-2(3H)-thiones, 1,3,4-oxadiazole-2(3H)-thiones, 4-amino-1,2,4-triazole-5(4H)-thiones, and substituted hydrazides to the dicopper active site

5. Structure activity studies of a novel cytotoxic benzodiazepine

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