Design, synthesis and evaluation of new 6-substituted-5-benzyloxy-4-oxo-4H-pyran-2-carboxamides as potential Src inhibitors-Reference-Cited by-同舟云学术

Design, synthesis and evaluation of new 6-substituted-5-benzyloxy-4-oxo-4H-pyran-2-carboxamides as potential Src inhibitors

Published:2008-01-01 Issue:5 Volume:23 Page:629-640
ISSN:1475-6366
Container-title:Journal of Enzyme Inhibition and Medicinal Chemistry
language:en
Short-container-title:Journal of Enzyme Inhibition and Medicinal Chemistry

Author:

Farard Julien¹,Lanceart Gaëtan¹,Logé Cedric¹,Nourrisson Marie-Renée¹,Cruzalegui Francisco²,Pfeiffer Bruno²,Duflos Muriel¹

Affiliation:

1. Département de Pharmacochimie, Faculté de Pharmacie, Université de Nantes, Nantes Atlantique UniversitésBioCiT-UPRES EA-1155, 1 rue Gaston Veil, NantesF-44035, France

2. Institut de Recherches Servier, 125 chemin de ronde, Croissy sur Seine 78290 France

Publisher

Informa UK Limited

Subject

Drug Discovery,Pharmacology,General Medicine

Link

https://www.tandfonline.com/doi/pdf/10.1080/14756360802205299

Reference20 articles.

1. Compensatory response to reducing body weight

2. Src inhibitors: drugs for the treatment of osteoporosis, cancer or both?

3. Role of Src expression and activation in human cancer

4. 2-Aminothiazole as a Novel Kinase Inhibitor Template. Structure−Activity Relationship Studies toward the Discovery of N-(2-Chloro-6-methylphenyl)-2-[[6-[4-(2-hydroxyethyl)-1- piperazinyl)]-2-methyl-4-pyrimidinyl]amino)]-1,3-thiazole-5-carboxamide (Dasatinib, BMS-354825) as a Potent pan-Src Kinase Inhibitor

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