Synthesis and Anti-HIV Activity of Some [Nucleoside Reverse Transcriptase Inhibitor]-C5′-Linker-[Integrase Inhibitor] Heterodimers as Inhibitors of HIV Replication-Reference-Cited by-同舟云学术

Synthesis and Anti-HIV Activity of Some [Nucleoside Reverse Transcriptase Inhibitor]-C5′-Linker-[Integrase Inhibitor] Heterodimers as Inhibitors of HIV Replication

Published:2004-12-01 Issue:6 Volume:19 Page:497-509
ISSN:1475-6366
Container-title:Journal of Enzyme Inhibition and Medicinal Chemistry
language:en
Short-container-title:Journal of Enzyme Inhibition and Medicinal Chemistry

Author:

Sugeac Elena¹,Fossey Christine¹,Ladurée Daniel¹,Schmidt Sylvie²,Laumond Geraldine²,Aubertin Anne-Marie²

Affiliation:

1. Centre d'Etudes et de Recherche sur le Médicament de Normandie, U.F.R. des Sciences Pharmaceutiques, 5, Rue Vaubénard, F-14032, Caen Cedex, France

2. I.N.S.E.R.M., 3, Rue Koeberlé, F-67000, Strasbourg, France

Publisher

Informa UK Limited

Subject

Drug Discovery,Pharmacology,General Medicine

Link

https://www.tandfonline.com/doi/pdf/10.1080/14756360412331280554

Reference35 articles.

1. AIDS — The challenge

2. Combination therapy for HIV-1 infection-overview: preclinical and clinical analysis of antiretroviral combinations

3. Toward Improved Anti-HIV Chemotherapy: Therapeutic Strategies for Intervention with HIV Infections

Cited by 4 articles. 订阅此论文施引文献订阅此论文施引文献，注册后可以免费订阅5篇论文的施引文献，订阅后可以查看论文全部施引文献

1. Polypharmacology in HIV inhibition: can a drug with simultaneous action against two relevant targets be an alternative to combination therapy?;European Journal of Medicinal Chemistry;2018-04

2. Synthesis of prodrug-type anti-HIV agents conjugating a REVERSE transcriptase inhibitor to a HIV-1 integrase inhibitor by a spontaneously cleavable linker;Journal of Enzyme Inhibition and Medicinal Chemistry;2007-01

3. Inhibitory activities against topoisomerase I & II by polyhydroxybenzoyl amide derivatives and their structure–activity relationship;Bioorganic & Medicinal Chemistry Letters;2004-04

4. Metabolites Produced by Actinomycetes-Antiviral Antibiotics and Enzyme Inhibitors-;YAKUGAKU ZASSHI;2004