Synthesis, characterization and preliminary screening of regioisomeric 1-(3-pyridazinyl)-3-arylpyrazole and 1-(3-pyridazinyl)-5-arylpyrazole derivatives towards cyclooxygenase inhibition-Reference-Cited by-同舟云学术

Synthesis, characterization and preliminary screening of regioisomeric 1-(3-pyridazinyl)-3-arylpyrazole and 1-(3-pyridazinyl)-5-arylpyrazole derivatives towards cyclooxygenase inhibition

Published:2007-01 Issue:3 Volume:22 Page:351-361
ISSN:1475-6366
Container-title:Journal of Enzyme Inhibition and Medicinal Chemistry
language:en
Short-container-title:Journal of Enzyme Inhibition and Medicinal Chemistry

Author:

Ünlü Serdar,Banoglu Erden,Ito Shigeru,Niiya Tokihiro,Eren Gökçen,Ökçelik Berna,Şahin Mustafa Fethi

Publisher

Informa UK Limited

Subject

Drug Discovery,Pharmacology,General Medicine

Link

http://www.tandfonline.com/doi/pdf/10.1080/14756360601073468

Reference34 articles.

1. Interpreting the clinical significance of the differential inhibition of cyclooxygenase-1 and cyclooxygenase-2

2. COX-2 Selectivity and Inflammatory Processes

3. Selective inhibition of inducible cyclooxygenase 2 in vivo is antiinflammatory and nonulcerogenic.

4. Cyclooxygenase-2 Inhibition and Side-effects of Non-steroidal Antiinflammatory Drugs in the Gastrointestinal Tract.

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