1. Synthesis of (+-)-7.beta.,8.alpha.-dihydroxy-9.beta.,10.beta.-epoxy-7,8,9,10-tetrahydrobenzo[a]pyrene, a potential metabolite of the carcinogen benzo[a]pyrene with stereochemistry related to the antileukemic triptolides
2. Tumorigenicity of the optical enantiomers of the diastereomeric benzo[a]pyrene 7,8-diol-9,10-epoxides in newborn mice: exceptional activity of (+)-7beta,8alpha-dihydroxy-9alpha,10alpha-epoxy-7,8,9,10-tetrahydrobenzo[a]pyrene.
3. Jerina, D. M., Sayer, J. M., Yagi, H., van Bladeren, P. J., Thakker, D. R., Levin, W., Chang, R. L., Wood, A. W. and Conney, A. H. 1985.Microsomes and Drug Oxidations, Edited by: Boobis, A. R., Caldwell, J., De Matteis, F. and Elcombe, C. R. 310–319. London: Taylor and Francis Ltd.
4. Dipple, A. 1994.DNA Adducts: Identification and Biological Significance, Edited by: Hemminki, K., Dipple, A., Shuker, D. E., Kadlubar, F. F., Segerback, D. and Bartsch, H. 107–129. Lyon: IARC Scientific Publication No. 125. b) D. M. Jerina, A. Chadha, A. M. Cheh, M. E. Schurdak, A. W. Wood and J. M. Sayer, inBiological Reactive Intermediates IV. Molecular and Cellular Effects and Their Impact on Human Health (Adv. Expt. Med. Biol.), edited by C. M. Witmer, R. Snyder, D. J. Jollow, G. F. Kalf, J. J. Kocsis and I. G. Sipes (Plenum Press, New York, 1991), pp. 533–553.
5. Lowry, T. H. and Richardson, K. S. 1976.Mechanism and Theory in Organic Chemistry, 149–150. New York: Harper and Row.