Quantification of osilodrostat in horse urine using LC/ESI–HRMS to establish an elimination profile for doping control

Author:

Ishii Hideaki12ORCID,Shigematsu Ryo1ORCID,Takemoto Shunsuke1,Ishikawa Yuhiro3,Mizobe Fumiaki3ORCID,Nomura Motoi3ORCID,Arima Daisuke4,Kunii Hirokazu4,Yuasa Reiko4,Yamanaka Takashi5,Tanabe Sohei5,Nagata Shun-ichi1,Yamada Masayuki1,Leung Gary Ngai-Wa1ORCID

Affiliation:

1. Drug Analysis Department, Laboratory of Racing Chemistry, 1731-2 Tsuruta-machi, Utsunomiya, Tochigi, 320-0851, Japan

2. Department of Pharmaceutical Sciences, Tohoku University Hospital, 1-1 Seiryo-machi, Aoba-ku, Sendai, Miyagi, 980-8574, Japan

3. Anti-Doping Section, Equine Department, Japan Racing Association, 1-1-1 Nishishimbashi, Minato-ku, Tokyo, 105-0003, Japan

4. Equine Veterinary Clinic, Horse Racing School, Japan Racing Association, 835-1 Ne Shiroi city, Chiba, Japan, 270-1431, Japan

5. Research Planning & Coordination Division, Equine Research Institute, Japan Racing Association, 1400-4 Shiba, Shimotsuke, Tochigi, 329-0412, Japan

Funder

The Japan Racing Association

Publisher

Informa UK Limited

Reference47 articles.

1. European Medicines Agency. Assessment report Isturisa [Internet]. Amsterdam: [updated 2019 November 14

2. cited 2024 May 15]. Available from: https://www.ema.europa.eu/en/documents/assessment-report/isturisa-epar-public-assessment-report_.pdf

3. Osilodrostat: First Approval

4. Annual banned‐substance review—Analytical approaches in human sports drug testing 2021/2022–

5. International Federation of Horseracing Authorities. International Agreement on Breeding Racing And Wagering And Appendixes (2023 edition with updated signatories) [Internet]. Paris: [updated 2024 May; cited 2024 May 15]. Available from: https://www.ifhaonline.org/resources/ifAgreement.pdf

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