1. The first reported observation of kinetic resolution: Pasteur ML (1858) C R Hebd Seances Acad Sci 46:615
2. (1) For a book and a review on α-hydroxy acids, see: (a) Coppola GM, Schuster HF (1997) α-Hydroxy acids in enantioselective syntheses. Wiley-VCH, Weinheim. (b) Gröger H (2001) Enzymatic Routes to Enantiomerically Pure Aromatic α‐Hydroxy Carboxylic Acids: A Further Example for the Diversity of Biocatalysis. Adv Synth Catal 343:547–558. (2) For the compounds described in Figure 2.3 (a) Evans JF, Kargman S (1992) Bestatin inhibits covalent coupling of [3H]LTA4 to human leukocyte LTA4hydrolase. FEBS Lett 297:139–142. (b) Tremblay LV, Xu H, Blanchard JS (2010) Structures of the Michaelis Complex (1.2 Å) and the Covalent Acyl Intermediate (2.0 Å) of Cefamandole Bound in the Active Sites of the Mycobacterium tuberculosis β-Lactamase K73A and E166A Mutants. Biochemistry 49:9685–9687. (c) Ebdrup S, Pettersson I, Rasmussen HB, Deussen HJ, Frost Jensen A, Mortensen SB, Fleckner J, Pridal L, Nygaard L, Sauerberg P (2003) Synthesis and Biological and Structural Characterization of the Dual-Acting Peroxisome Proliferator-Activated Receptor α/γ Agonist Ragaglitazar. J Med Chem 46:1306–1317
3. (a) Gao Y, Hanson RM, Klunder JM, Ko SY, Masamune H, Sharpless KB (1987) Catalytic asymmetric epoxidation and kinetic resolution: modified procedures including in situ derivatization. J Am Chem Soc 109:5765-5780.
4. (b) Bauer T, Tarasiuk J (2002) α-Hydroxy carboxylic acids: new ligands for diethylzinc additions to aldehydes. Tetrahedron Lett 43:687-689.
5. (c) Bauer T, Gajewiak J (2004) α-Hydroxy carboxylic acids as ligands for enantioselective diethylzinc additions to aromatic and aliphatic aldehydes. Tetrahedron 60:9163-9170.