Binding of the A1-selective adenosine antagonist 8-cyclopentyl-1,3-dipropylxanthine to rat brain membranes

Author:

Bruns Robert F.,Fergus James H.,Badger Edward W.,Bristol James A.,Santay Lisa A.,Hartman Jon D.,Hays Sheryl J.,Huang Che C.

Publisher

Springer Science and Business Media LLC

Subject

Pharmacology,General Medicine

Reference21 articles.

1. Blicke FF, Godt HC Jr (1954) Reactions of 1,3-dimethyl-5,6-diaminouracil. J Am Chem Soc 76:2798?2800

2. Bruns RF, Daly JW, Snyder SH (1980) Adenosine receptors in brain membranes: Binding of N6-cyclohexyl[3H]adenosine and 1,3-diethyl-8-[3H]phenylxanthine. Proc Natl Acad Sci USA 77: 5547?5551

3. Bruns RF, Daly JW, Snyder SH (1983) Adenosine receptor binding: Structure-activity analysis generates extremely potent xanthine antagonists. Proc Natl Acad Sci USA 80:2077?2080

4. Bruns RF, Lu GH, Pugsley TA (1984) Binding of 3H-NECA to a subtype of A2 adenosine receptor in rat striatal membranes. Soc Neurosci Abstr 10:957

5. Bruns RF, Lu GH, Pugsley TA (1985) Towards selective adenosine antagonists. In: Stefanovich V, Rudolphi K, Schubert P (eds) Adenosine: Receptors and modulation of cell functions. IRL Press, Oxford, pp 51?58

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