5-HT1A receptor pharmacophores to screen for off-target activity of α1-adrenoceptor antagonists-Reference-Cited by-同舟云学术

5-HT1A receptor pharmacophores to screen for off-target activity of α1-adrenoceptor antagonists

Published:2013-04 Issue:4 Volume:27 Page:305-319
ISSN:0920-654X
Container-title:Journal of Computer-Aided Molecular Design
language:en
Short-container-title:J Comput Aided Mol Des

Author:

Ngo Tony,Nicholas Timothy J.,Chen Junli,Finch Angela M.,Griffith Renate

Publisher

Springer Science and Business Media LLC

Subject

Physical and Theoretical Chemistry,Computer Science Applications,Drug Discovery

Link

http://link.springer.com/content/pdf/10.1007/s10822-013-9647-5.pdf

Reference78 articles.

1. Guiard BP, El Mansari M, Merali Z, Blier P (2008) Functional interactions between dopamine, serotonin and norepinephrine neurons: an in vivo electrophysiological study in rats with monoaminergic lesions. Int J Neuropsychoph 11(5):625–639

2. Kenakin T (2010) A holistic view of GPCR signaling. Nat Biotechnol 28(9):928–929

3. Ahmad N, Keith-Ferris J, Gooden E, Abell T (2006) Making a case for domperidone in the treatment of gastrointestinal motility disorders. Curr Opin Pharmacol 6(6):571–576

4. Albert PR, Zhou QY, Vantol HHM, Bunzow JR, Civelli O (1990) Cloning, functional expression, and messenger-RNA tissue distribution of the rat 5-hydroxytryptamine-1a receptor gene. J Biol Chem 265(10):5825–5832

5. Gitler MS, Piccio MM, Robillard JE, Jose PA (1991) Characterization of renal alpha-adrenoceptor subtypes in sheep during development. Am J Physiol 260(2):R407–R412

Cited by 9 articles. 订阅此论文施引文献订阅此论文施引文献，注册后可以免费订阅5篇论文的施引文献，订阅后可以查看论文全部施引文献

1. New Serotoninergic Ligands Containing Indolic and Methyl Indolic Nuclei: Synthesis and In Vitro Pharmacological Evaluation;Medicinal Chemistry;2020-05-20

2. Synthesis, in vitro and in vivo evaluation of 11C-O-methylated arylpiperazines as potential serotonin 1A (5-HT1A) receptor antagonist radiotracers;EJNMMI Radiopharmacy and Chemistry;2020-05-19

3. In Silico Studies Targeting G-protein Coupled Receptors for Drug Research Against Parkinson’s Disease;Current Neuropharmacology;2018-06-08

4. Pharmacophore Models for Toxicology Prediction;Computational Toxicology;2018-01-19

5. Synthesis and activity of newly designed aroxyalkyl or aroxyethoxyethyl derivatives of piperazine on the cardiovascular and the central nervous systems;Bioorganic & Medicinal Chemistry Letters;2016-11