The efficacy of selinexor (KPT-330), an XPO1 inhibitor, on non-hematologic cancers: a comprehensive review

Author:

Landes Jennifer R.ORCID,Moore Stephen A.,Bartley Brooke R.,Doan Hung Q.,Rady Peter L.,Tyring Stephen K.

Publisher

Springer Science and Business Media LLC

Subject

Cancer Research,Oncology,General Medicine

Reference97 articles.

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2. Aboukameel A, Muqbil I, Baloglu E, Senapedis W, Landesman Y, Argueta C, Kauffman M, Chang H, Kashyap T, Shacham S, Neggers JE, Daelemans D, Heath EI, Azmi AS (2018) Down-regulation of AR splice variants through XPO1 suppression contributes to the inhibition of prostate cancer progression. Oncotarget. https://doi.org/10.18632/oncotarget.26239

3. Aladhraei M, Kassem Al-Thobhani A, Poungvarin N, Suwannalert P (2019) Association of XPO1 Overexpression with NF-κB and Ki67 in colorectal cancer. Asian Pac J Cancer Prev 20(12):3747–3754. https://doi.org/10.31557/apjcp.2019.20.12.3747

4. Alzahrani A, Natarajan U, Rathinavelu A (2022) Enhancement of MDM2 inhibitory effects through blocking nuclear export mechanisms in ovarian cancer cells. Cancer Genet 266–267:57–68. https://doi.org/10.1016/j.cancergen.2022.06.003

5. Arango NP, Yuca E, Zhao M, Evans KW, Scott S, Kim C, Gonzalez-Angulo AM, Janku F, Ueno NT, Tripathy D, Akcakanat A, Naing A, Meric-Bernstam F (2017) Selinexor (KPT-330) demonstrates anti-tumor efficacy in preclinical models of triple-negative breast cancer. Breast Cancer Res 19(1):93. https://doi.org/10.1186/s13058-017-0878-6

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