Phosphinic Dehydrodipeptides: Diversification of the P1′ Residue with the Morita–Baylis–Hillman Acetates and Inhibition of Alanyl Aminopeptidases
Author:
Funder
Narodowe Centrum Nauki
Publisher
Springer Science and Business Media LLC
Subject
Drug Discovery,Molecular Medicine,Biochemistry,Bioengineering,Analytical Chemistry
Link
http://link.springer.com/content/pdf/10.1007/s10989-019-10004-7.pdf
Reference34 articles.
1. Basavaiah D, Pandiaraju S (1996) Nucleophilic addition of triethyl phosphite to acetates of the Baylis–Hillman adducts: stereoselective synthesis of (E)- and (Z)-allylphosphonates. Tetrahedron 52:2261–2268. https://doi.org/10.1016/0040-4020(95)01055-6
2. Baylis EK, Campbell CD, Dingwall JG (1984) 1-Aminoalkylphosphonous acids. Part 1. Isosteres of the protein amino acids. J Chem Soc Perkin Trans 1:2845–2853. https://doi.org/10.1039/P19840002845
3. Boyd EA, Corless M, James K, Regan AC (1990) A versatile route to substituted phosphinic acids. Tetrahedron Lett 31:2933–2936. https://doi.org/10.1016/0040-4039(90)80188-R
4. Chen H, Noble F, Mothé A, Hervé M, Coric P, Danascimento S, Roques BP, George P, Fournié-Zaluski MC (2000) Phosphinic derivatives as new dual enkephalin-degrading enzyme inhibitors: synthesis, biological properties, and antinociceptive activities. J Med Chem 43:1398–1408. https://doi.org/10.1021/jm990483l
5. Chen S, Coward JK (1996) A general method for the synthesis of N-protected α-aminoalkylphosphinic acids. Tetrahedron Lett 37:4335–4338. https://doi.org/10.1016/0040-4039(96)00839-8
Cited by 3 articles. 订阅此论文施引文献 订阅此论文施引文献,注册后可以免费订阅5篇论文的施引文献,订阅后可以查看论文全部施引文献
1. Inhibition of glutathione S-transferases by calix[4]arene-based phosphinic acids;Ukr. Bioorg. Acta 2022, Vol. 17, N1;2022-06-30
2. P1′ Residue-Oriented Virtual Screening for Potent and Selective Phosphinic (Dehydro) Dipeptide Inhibitors of Metallo-Aminopeptidases;Biomolecules;2020-04-24
3. Synthesis and Structure-Activity Relationship Studies of Hydrazide-Hydrazones as Inhibitors of Laccase from Trametes versicolor;Molecules;2020-03-10
1.学者识别学者识别
2.学术分析学术分析
3.人才评估人才评估
"同舟云学术"是以全球学者为主线,采集、加工和组织学术论文而形成的新型学术文献查询和分析系统,可以对全球学者进行文献检索和人才价值评估。用户可以通过关注某些学科领域的顶尖人物而持续追踪该领域的学科进展和研究前沿。经过近期的数据扩容,当前同舟云学术共收录了国内外主流学术期刊6万余种,收集的期刊论文及会议论文总量共计约1.5亿篇,并以每天添加12000余篇中外论文的速度递增。我们也可以为用户提供个性化、定制化的学者数据。欢迎来电咨询!咨询电话:010-8811{复制后删除}0370
www.globalauthorid.com
TOP
Copyright © 2019-2024 北京同舟云网络信息技术有限公司 京公网安备11010802033243号 京ICP备18003416号-3