Synthesis of new chiral 1,3,4-thiadiazole-based di- and tri-arylsulfonamide residues and evaluation of in vitro anti-HIV activity and cytotoxicity-Reference-Cited by-同舟云学术

Synthesis of new chiral 1,3,4-thiadiazole-based di- and tri-arylsulfonamide residues and evaluation of in vitro anti-HIV activity and cytotoxicity

Published:2018-07-02 Issue:4 Volume:22 Page:957-968
ISSN:1381-1991
Container-title:Molecular Diversity
language:en
Short-container-title:Mol Divers

Author:

Shafique Maria,Hameed Shahid,Naseer Muhammad Moazzam,Al-Masoudi Najim Aboud

Publisher

Springer Science and Business Media LLC

Subject

Inorganic Chemistry,Organic Chemistry,Physical and Theoretical Chemistry,Drug Discovery,Molecular Biology,General Medicine,Information Systems,Catalysis

Link

http://link.springer.com/article/10.1007/s11030-018-9851-2/fulltext.html

Reference44 articles.

1. Li Y, Geng J, Liu Y, Yu S, Zhao G (2013) Thiadiazole a promising structure in medicinal chemistry. ChemMedChem 8:27–41. https://doi.org/10.1002/cmdc.201200355

2. Hu Y, Li C-Y, Wang X-M, Yang Y-H, Zhu H-L (2014) 1,3,4-Thiadiazole: synthesis, reactions, and applications in medicinal, agricultural, and materials chemistry. Chem Rev 114:5572–5610. https://doi.org/10.1021/cr400131u

3. Jain AK, Sharma S, Vaidya A, Ravichandran V, Agrawal RK (2013) 1,3,4-Thiadiazole and its derivatives: a review on recent progress in biological activities. Chem Biol Drug Des 81:557–576. https://doi.org/10.1111/cbdd.12125

4. Ezabadi IR, Camoutsis C, Zoumpoulakis P, Geronikaki A, Soković M, Glamocilija J, Cirić A (2008) Sulfonamide-1,2,4-triazole derivatives as antifungal and antibacterial agents: synthesis, biological evaluation, lipophilicity, and conformational studies. Bioorg Med Chem 16:1150–1161. https://doi.org/10.1016/j.bmc.2007.10.082

5. Kumura K, Wakiyama Y, Ueda K, Umemura E, Watanabe Yamamoto M, Yoshida T, Ajito K (2018) Synthesis and antibacterial activity of novel lincomycin derivatives. III. Optimization of a phenyl thiadiazole moiety. J Antibiot 71:104–112. https://doi.org/10.1038/ja.2017.59

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